
李晓婷,1989年10月生,陕西省定边人,沈阳药科大学理学博士,延边大 学药学院副教授,硕士研究生导师,《亚洲药物制剂科学》青年编委。主持国 家自然科学基金(青年基金)1项,吉林省自然科学基金1项,省教育厅项目1项, 图们江计划2项,省级教研项目1项,校级项目3项。以第一或者通讯作者发表二 区以上SCI论文十余篇,其中Eur J Med Chem 、Molecular Pharmaceutics 等国际 药学Top期刊上发表8篇高水平SCI论文,申请专利2项。获吉林省高层次E类人才、 青年图们江学者、青年图们江学者B类(人才引进)、吉林省“建行杯 ”第八届 “互联网+ ”大学生创新创业大赛铜奖指导教师奖、吉林省第四届“超星杯 ”高 校教师教学创新大赛一等奖等荣誉。
【联系方式】0433-2732134;15524295943;E-mail: sypulixiaoting@163.com
【研究方向】1.基于代谢酶/转运体的前药设计与评价;
2.基于生理药动学模型的药物相互作用研究;
3.体内药物分析新技术与方法研究。
【主持科研项目】
1.双重评估预测质子泵抑制剂与pH-依赖型BCS2 类药物相互作用的药动学 模 型研究,国家自然科学基金(82204310),2023-2025 ,30 万,在研,主持。
2.In-silico/In-vitro 偶联 GIS-PBPK 模型助力 BCSII 类弱酸性 NSAIDs 仿制 药 一致性评,吉林省自然科学基金(YDZJ202301ZYTS143), 2023--2025, 10 万, 在研,主持。
3.基于 GIS 偶联 PBPK 模型定量研究 PPIs 对萘普生药动学的影响,吉林省 教 育厅项目(JJKH20220563KJ), 2021-01-2023-12, 2.5 万,在研,主持。
4.以就业为导向的“产教融合—拔尖创新型 ”药学人才培养模式研究(GH24380) ,药学“专业教育 ”吉林省教育科学“十四五 ”规划课题,20241019- 20261019,1.0万,在研,主持。
【代表性论文】
(1) Dan Wu 1, Xiaoting Li 1, Qing-Kun Shen, Run-Hui Zhang, Qian Xu, Xiao-Tong Sang, Xing Huang, Chang-Hao Zhang, Zhe-Shan Quan, Li-Hua Cao, Design, synthesis and biological evaluation of dehydroabietic acid derivative as potent vasodilatory agents, Bioorganic Chemistry, 2022, 129: 106110. (SCI 1 区,并列 一作)
(2) Fan-Fan Shang, Jing Ying Wang, Qian Xu, Hao Deng, Hong-Yan Guo, Xuejun Jin, Xiaoting Li*, Qing-Kun Shen*, Zhe-Shan Quan*. Design, synthesis of novel celastrol derivatives and study on their antitumor growth through HIF-1a pathway ,Eur JMed Chem, 2021, 220:113474. (SCI 1 区)
(3) Hong-Yan Guo1, Xiaoting Li1, Xiao-Tong Sang , Zhe-Shan Quan *, Qing-Kun Shen **. Design and synthesis of forsythin derivatives as anti-inflammatory agents for acute lung injury. Eur JMed Chem, 2024, 267: 116223. (SCI 1 区)
(4) Miao-Xia Pu, Hong-Yan Guo, Zhe-Shan Quan, Xiaoting Li* and Qing-Kun Shen*, Application of the Mannich reaction in the structural modification of natural products.JournalofEnzyme i ition CInhbandMedicinalhemistry, 2023 , 38(1): 2235095 (SCI 2 区)
(5) Xing Huang, Qing-Kun Shen, Hong-Yan Guo, Zhe-Shan Quan*, Xiaoting Li*,Research, development and pharmacological activity of fusidic acid and its derivatives, Journal ofMolecular Structure, 2023, 1291: 135942. (SCI 2 区)
(6) Jin-Ying Liu, Hong-Yan Guo, Zhe-Shan Quan, Qing-Kun Shen, Hong Cui and Xiaoting Li*, Research progress of natural products and their derivatives against Alzheimer ’sdisease,Journal ofEnzyme Inhibition and Medicinal Chemistry, 2023, 38(1): 2171026. (SCI 2 区)
(7) Qian Xu, Hao Deng, Xiaoting Li*, Zhe-Shan Quan*, Application of Amino Acids in the Structural Modification of Natural Products: A Review, Frontiers in Chemistry, 2021, 9: 650569. (SCI 2 区)
(8) Xiaoting Li, Yuanhang Yang,Yu Zhang,Chunnuan Wu,Qikun Jiang,Weiping Wang,Huixin Li,Jing Li,Cong Luo,Wenying, Yingli Wang , Tianhong Zhang, Justification of Biowaiver and Dissolution Rate Specifications for Piroxicam Immediate Release Products Based on Physiologically Based Pharmacokinetic Modeling: An In-Depth Analysis,Mol. Pharmaceutics, 2019, 16, (9): 3780 -3790. (SCI 2 区)